Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_03805
Ion Channel
Sodium channel type 8 subunit alpha
Peptide Function
Blocker
Gene Name
Scn8a
Activity Data (nM)
IC50
Not available
Ki
Not available
EC50
2265 nM
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
GTPCYCGKTIGIYWFGTKTCPSNRGYTGSCGYFLGICCYPVD
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
APETx3
Peptide Species
Anthopleura elegantissima (Green aggregating anemone) (Actinia elegantissima)
Peptide Name
Delta-actitoxin-Ael2d
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−90 mV
Temperature
18–22 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Mus musculus (Mouse)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available